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Advanced Pharmaceutical Solids
1. One Component System...1
2. Properties of Solids...13
3. Solubility...27
4. Particle Sixes and Diameters...51
5. Micromeritics...61
6. Crystalization...89
7. Amorphates...107
8. Polymorphism...117
9. Moisture Isotherms with Crystalline Solids...133
10. Drug Substance Considerations...159
11. Melting Point Diagrams and Eutetics...169
12. Dissolution From Particles and Surfaces...191
13. Dissolution from Polydisperse Populations...209
14. Solid State Stability...223
15. Effect of Moisture on Solid-State Stability...267
16. Apparent Volumes and Densities...281
17. Cohesion...299
18. Powder Flow...309
19. Comminution...323
20. Blending...335
21. Wet Granulation...353
22. Hard Shell Capsules..375
23. Tablet Physic...387
24. Physical Principles of Tablets...407
25. Disintegration and Dissolution...427
26. Polymers...439
27. Coating of Tablets...455
28. Single Unit Sustained Release Dosage Forms...469
29. Sustained Release by Microencapsulation...493
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